SCHEMBL28620218

SCHEMBL28620218

COc1ccc(COC2CCc3ccc(CO)cc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.43
BRD4 O60885 1/20 0.43
CYP24A1 Q07973 1/20 0.41
MTNR1A P48039 7/20 0.41
NQO2 P16083 6/20 0.39
MTNR1B P49286 6/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
CYP3A4 P08684 1/20 0.39
STS P08842 1/20 0.39
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20241215 0.84 BRD4 (0.43) CYP26A1BRD4CYP24A1MTNR1AMAPT
SCHEMBL18322124 0.81 NPC1 (0.48) CYP26A1BRD4CYP24A1MTNR1ANQO2
SCHEMBL28615795 0.78 THRB (0.50) CYP26A1BRD4CYP24A1KDM4EMAPT
SCHEMBL18322201 0.78 THRB (0.50) CYP26A1BRD4CYP24A1KDM4EMAPT
SCHEMBL5206057 0.78 MAOB (0.42) CYP26A1BRD4CYP24A1MAPTSTS
SCHEMBL18322205 0.77 NR1H4 (0.47) MTNR1ANQO2MTNR1BKDM4EMAPT
SCHEMBL20241344 0.77 NR1H4 (0.47) MTNR1ANQO2MTNR1BKDM4EMAPT
SCHEMBL18321967 0.74 MTNR1A (0.37) MTNR1ANQO2MTNR1BALDH1A1
SCHEMBL18321982 0.73 FFAR1 (0.41) CYP26A1BRD4CYP24A1
SCHEMBL18321978 0.73 BRD4 (0.38) CYP26A1BRD4CYP24A1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137557-B Nrf2 modulators 葛兰素史密斯克莱知识产权发展有限公司 2021-09-07 CN disclosed