SCHEMBL28620280

SCHEMBL28620280

C=CC(=O)Nc1ccc(C(=O)N[C@@H](C)c2ccc(F)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 3/20 0.61
NPC1 O15118 3/20 0.60
KMT2A Q03164 4/20 0.59
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
MEN1 O00255 2/20 0.51
HTT P42858 2/20 0.51
PTPN1 P18031 1/20 0.46
CTNNB1 P35222 2/20 0.45
TCF7L2 Q9NQB0 2/20 0.45
RAB9A P51151 2/20 0.45
NR1H4 Q96RI1 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ROCK2 O75116 1/20 0.45
ATM Q13315 1/20 0.45
MITF O75030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28619301 1.00 TGM2 (0.61) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28617576 0.88 TGM2 (0.66) TGM2NPC1KMT2AMEN1RAB9A
SCHEMBL28615912 0.87 TGM2 (0.61) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28624100 0.87 B3GNT2 (0.47) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28627367 0.87 TGM2 (0.47) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28630813 0.87 KMT2A (0.60) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28619644 0.87 KMT2A (0.60) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28617369 0.87 KMT2A (0.60) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28616230 0.85 NPC1 (0.52) TGM2NPC1KMT2AALDH1A1LMNA
SCHEMBL28615353 0.85 TGM2 (0.66) TGM2NPC1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438279-B Small molecule compound for overcoming EGFR drug-resistant mutation and preparation method and application thereof 四川大学 2021-08-31 CN disclosed