SCHEMBL28615353

SCHEMBL28615353

C=CC(=O)Nc1ccc(C(=O)N[C@@H](C)c2ccc(OC)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.66
TAS1R3 Q7RTX0 1/20 0.54
TAS1R1 Q7RTX1 1/20 0.54
RAB9A P51151 6/20 0.54
NPC1 O15118 5/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TP53 P04637 1/20 0.54
ALOX15 P16050 1/20 0.54
CNR1 P21554 2/20 0.53
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
LMNA P02545 2/20 0.48
PKM P14618 1/20 0.48
OPRD1 P41143 1/20 0.48
F2 P00734 1/20 0.47
F10 P00742 1/20 0.47
F7 P08709 1/20 0.47
MAPT P10636 3/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28619301 0.85 TGM2 (0.61) TGM2RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL28624100 0.85 B3GNT2 (0.47) TGM2RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL28627367 0.85 TGM2 (0.47) TGM2NPC1SMN1; SMN2TP53MEN1
SCHEMBL28620280 0.85 TGM2 (0.61) TGM2RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL28615912 0.85 TGM2 (0.61) TGM2RAB9ANPC1SMN1; SMN2CNR1
SCHEMBL28617369 0.85 KMT2A (0.60) TGM2NPC1SMN1; SMN2TP53MEN1
SCHEMBL28619644 0.85 KMT2A (0.60) TGM2NPC1SMN1; SMN2TP53MEN1
SCHEMBL28630813 0.85 KMT2A (0.60) TGM2NPC1SMN1; SMN2TP53MEN1
SCHEMBL28354065 0.84 TAS1R3 (0.70) TAS1R3TAS1R1RAB9ANPC1SMN1; SMN2
SCHEMBL28617576 0.83 TGM2 (0.66) TGM2RAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438279-B Small molecule compound for overcoming EGFR drug-resistant mutation and preparation method and application thereof 四川大学 2021-08-31 CN disclosed