SCHEMBL28622709

SCHEMBL28622709

CCOC(=O)C(N)Cc1ccc(OC)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
SCN9A Q15858 1/20 0.47
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
HTR2A P28223 1/20 0.46
APLNR P35414 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23201898 0.89 APLNR (0.51) ALDH1A1POLBHTR2AAPLNRDPP7
SCHEMBL23201900 0.89 APLNR (0.51) ALDH1A1POLBHTR2AAPLNRDPP7
SCHEMBL491054 0.86 ALDH1A1 (0.51) ALDH1A1POLBTDP1TSHRMAPK1
SCHEMBL29519833 0.84 HSD17B10 (0.49) ALDH1A1POLBTDP1HTR2AAPLNR
Hydrochloric Acid SCHEMBL8862614 0.83 HSD17B10 (0.48) HTR2AAPLNRDPP7MEN1KMT2A
SCHEMBL20543840 0.81 ALDH1A1 (0.47) ALDH1A1POLBSCN9ATSHRMEN1
SCHEMBL26985715 0.81 ALDH1A1 (0.47) ALDH1A1POLBSCN9ATSHRMEN1
SCHEMBL6301729 0.80 SCN9A (0.60) SCN9AHTR2AMEN1KMT2AMAPT
SCHEMBL21384322 0.80 SCN9A (0.60) SCN9AHTR2AMEN1KMT2AMAPT
SCHEMBL17500269 0.80 SCN9A (0.69) ALDH1A1TDP1SCN9ATSHRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115485276-B Deuterated AKT kinase inhibitors 南京正大天晴制药有限公司 2024-05-31 CN disclosed
CN-117964620-A AKT inhibitors 南京正大天晴制药有限公司 2024-05-03 CN disclosed
CN-113272304-B AKT inhibitors 南京正大天晴制药有限公司 2024-03-29 CN disclosed
CN-115485276-A Deuterated AKT kinase inhibitors 南京正大天晴制药有限公司 2022-12-16 CN disclosed
CN-113272304-A AKT inhibitors 南京正大天晴制药有限公司 2021-08-17 CN disclosed