SCHEMBL28623966

SCHEMBL28623966

CC(=O)c1ccc(C)cc1NC(=O)c1ccccn1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.65
NPC1 O15118 4/20 0.65
RAB9A P51151 4/20 0.65
NFKB1 P19838 2/20 0.65
NFKB2 Q00653 2/20 0.65
RELA Q04206 2/20 0.65
GAA P10253 2/20 0.65
KDR P35968 1/20 0.55
HTT P42858 3/20 0.55
OPRK1 P41145 1/20 0.55
GRM4 Q14833 2/20 0.53
LMNA P02545 2/20 0.52
ALDH1A1 P00352 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KMT2A Q03164 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29643961 1.00 MAPT (0.65) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL28620094 0.89 NPC1 (0.69) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL29643911 0.89 NPC1 (0.69) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL29644052 0.86 GRM4 (0.59) NPC1RAB9AKDRGRM4KMT2A
SCHEMBL28628481 0.86 GRM4 (0.59) NPC1RAB9AKDRGRM4KMT2A
SCHEMBL31087264 0.84 HDAC6 (0.62) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL28611795 0.84 HDAC6 (0.62) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL1536653 0.83 RAB9A (0.65) MAPTNPC1RAB9AHTTGRM4
SCHEMBL29644059 0.78 GRM4 (0.59) MAPTNPC1RAB9ANFKB1NFKB2
SCHEMBL28625315 0.78 GRM4 (0.59) MAPTNPC1RAB9ANFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113278007-B Synthetic method of 2-hydroxy-indole-3-ketone compound 延安大学 2022-05-17 CN disclosed
CN-113278007-A Synthetic method of 2-hydroxy-indole-3-ketone compound 延安大学 2021-08-20 CN disclosed