SCHEMBL2862398

SCHEMBL2862398

O=S(=O)(c1ccccc1)c1cc(O)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 1.00
POLB P06746 2/20 1.00
GFER P55789 2/20 1.00
TDP1 Q9NUW8 2/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
ALPL P05186 1/20 0.61
ALPI P09923 1/20 0.61
ALPG P10696 1/20 0.61
DNMT1 P26358 1/20 0.61
MCL1 Q07820 1/20 0.61
ALDH1A1 P00352 1/20 0.60
PKM P14618 1/20 0.60
PTGS1 P23219 1/20 0.53
ATM Q13315 2/20 0.53
ERAP1 Q9NZ08 2/20 0.53
HTR6 P50406 2/20 0.48
MEN1 O00255 1/20 0.47
PABPC1 P11940 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10489216 0.90 GAA (0.81) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL8526863 0.87 GAA (0.77) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL6534882 0.85 GAA (0.73) GAAPOLBGFERL3MBTL1ALDH1A1
SCHEMBL660467 0.85 GAA (0.73) GAAPOLBGFERL3MBTL1ALDH1A1
SCHEMBL979753 0.85 POLB (0.73) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL900962 0.83 ALPL (0.74) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL30678705 0.83 ALPL (0.74) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL9001240 0.81 GAA (0.69) GAAPOLBGFERL3MBTL1ALDH1A1
SCHEMBL4961422 0.81 POLB (0.70) GAAPOLBGFERTDP1L3MBTL1
SCHEMBL17774551 0.81 POLB (0.69) GAAPOLBGFERTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4814416-A SULFONE CONTAINING DIOLS HUELS AKTIENGESELLSCHAFT (DE) 1989-03-21 US claimed
EP-0203468-B1 IMPROVED PHOTOGRAPHIC MATERIAL FOR TANNING DEVELOPMENT AND METHOD FOR OBTAINING A RELIEF IMAGE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1989-03-08 EP claimed
US-4737441-A INCLUDING TWO DIFFERENT SUBSTITUTED 1,4-DIHYDRONBENZENES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1988-04-12 US claimed
EP-0203468-A2 Improved photographic material for tanning development and method for obtaining a relief image MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1986-12-03 EP claimed
US-7713449-B2 Polymer electrolytic material, polymer electrolytic part, membrane electrode assembly, and polymer electrolyte fuel cell TORAY INDUSTRIES, INC. (JP) 2010-05-11 US disclosed
US-20070173548-A1 Malonamic acids and derivatives thereof as thyroid receptor ligands CHIANG YUAN-CHING P 2007-07-26 US disclosed
US-7202275-B2 Malonamic acids and derivatives thereof as thyroid receptor ligands WARNER LAMBERT COMPANY LLC (US) 2007-04-10 US disclosed
US-20060180796-A1 Polymer electrolyte material, polymer electrolyte part, membrane electrode composite and polymer electrolyte type fuel cell TORAY INDUSTRIES, INC. (JP) 2006-08-17 US disclosed
CN-1757130-A Polymer electrolyte material, polymer electrolyte part, film electrode composite element and polymer electrolyte fuel cells TORAY INDUSTRIES (JP) 2006-04-05 CN disclosed
EP-1619735-A1 POLYMER ELECTROLYTE MATERIAL, POLYMER ELECTROLYTE PART, MEMBRANE ELECTRODE COMPOSITE AND POLYMER ELECTROLYTE TYPE FUEL CELL TORAY INDUSTRIES, INC. (JP) 2006-01-25 EP disclosed
WO-2002090344-A1 AMIDO-DIPHENYL DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2002-11-14 WO disclosed
EP-0662004-B1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1998-03-18 EP disclosed
EP-0501922-A2 Compositions based on polyamide-polyimide block copolymers CIBA-GEIGY AG (CH) 1992-09-02 EP disclosed
US-4814416-A SULFONE CONTAINING DIOLS HUELS AKTIENGESELLSCHAFT (DE) 1989-03-21 US disclosed
EP-0203468-B1 IMPROVED PHOTOGRAPHIC MATERIAL FOR TANNING DEVELOPMENT AND METHOD FOR OBTAINING A RELIEF IMAGE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1989-03-08 EP disclosed
US-4752547-A RECORDING LAYER CONTAINS REDUCING AGENT, LEWIS BASE COMPLEX, AND REDUCIBLE DYE FORMING COMPOUND EASTMAN KODAK COMPANY (US) 1988-06-21 US disclosed
US-4737441-A INCLUDING TWO DIFFERENT SUBSTITUTED 1,4-DIHYDRONBENZENES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1988-04-12 US disclosed
US-4727008-A MULTILAYER-IMAGEWISE EXPOSURE TO ELECTRICAL CHARGES OF DIFFERENT POLARITIES TO GIVE DEVELOPABLE IMAGES EASTMAN KODAK COMPANY (US) 1988-02-23 US disclosed
EP-0203468-A2 Improved photographic material for tanning development and method for obtaining a relief image MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1986-12-03 EP disclosed
US-4299946-A THERMOSETTING RESINS RHONE-POULENC INDUSTRIES (FR) 1981-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070173548-A1 Malonamic acids and derivatives thereof as thyroid receptor ligands THRA, MC1R, TSHR GAA 521/4885POLB 1875/4885GFER 2519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.