SCHEMBL28625832

SCHEMBL28625832

COc1cccc2cc(C(=O)NNC(=O)Nc3ccc(CN4CCC(C)CC4)cc3)c(=O)oc12

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
HSD17B10 Q99714 2/20 0.60
HPGD P15428 2/20 0.60
MAPT P10636 3/20 0.57
TP53 P04637 1/20 0.57
BACE1 P56817 1/20 0.54
POLB P06746 3/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 3/20 0.50
RXFP1 Q9HBX9 2/20 0.50
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641065 0.93 TP53 (0.67) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28621577 0.90 POLB (0.46) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28621580 0.85 ALDH1A1 (0.52) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28636610 0.82 AKR1C3 (0.52) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28626014 0.81 MAPT (0.65) ALDH1A1HSD17B10MAPTTP53POLB
SCHEMBL28625763 0.80 MAPT (0.62) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28630602 0.79 HPGD (0.53) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL28629444 0.76 CASP3 (0.53) ALDH1A1HSD17B10HPGD
SCHEMBL28641067 0.73 MAPT (0.76) ALDH1A1HSD17B10MAPTTP53POLB
SCHEMBL981812 0.71 MAPT (0.78) ALDH1A1HSD17B10MAPTTP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108715589-B Coumarin derivative used as caspase-3 activator and application thereof 华侨大学 2021-04-20 CN disclosed