SCHEMBL28625906

SCHEMBL28625906

O=C(O)C(COc1cccc(Cl)c1)NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
ALOX12 P18054 1/20 0.43
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
PKM P14618 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30854486 1.00 RXRA (0.43) RXRARXRBRXRGTP53GAA
SCHEMBL21837588 0.89 KDM4E (0.43) RXRARXRBRXRGKDM4EPKM
SCHEMBL17491917 0.89 KDM4E (0.43) RXRARXRBRXRGKDM4EPKM
SCHEMBL17491919 0.89 KDM4E (0.43) RXRARXRBRXRGKDM4EPKM
SCHEMBL7656116 0.87 MTNR1A (0.45) CYP2D6
SCHEMBL7656123 0.87 MTNR1A (0.45) CYP2D6
SCHEMBL16094419 0.85 HTT (0.47) KDM4E
SCHEMBL16094416 0.85 HTT (0.47) KDM4E
SCHEMBL19377978 0.81 SMN1; SMN2 (0.52) TP53NPC1RAB9APKM
SCHEMBL19377976 0.81 SMN1; SMN2 (0.52) TP53NPC1RAB9APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118256591-A Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-06-28 CN disclosed
CN-118184532-A Amino acid having functional group capable of forming intramolecular hydrogen bond, peptide compound containing the amino acid, and process for producing the same 中外制药株式会社 2024-06-14 CN disclosed
CN-113454058-B Amino acid having functional group capable of forming intramolecular hydrogen bond, peptide compound containing the amino acid, and process for producing the same 中外制药株式会社 2024-03-22 CN disclosed
CN-110869544-B Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-03-08 CN disclosed
CN-113454058-A Amino acid having functional group capable of forming intramolecular hydrogen bond, peptide compound comprising the same, and method for producing the same 中外制药株式会社 2021-09-28 CN disclosed