SCHEMBL28626909

SCHEMBL28626909

COC(=O)CCc1c(C)n(C)c2ccc(C(F)(F)F)cc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.47
SPR P35270 1/20 0.47
TACR1 P25103 1/20 0.41
SRC P12931 1/20 0.41
AKR1C2 P52895 2/20 0.41
KIF11 P52732 1/20 0.40
CYP2C9 P11712 1/20 0.40
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
PTGDR2 Q9Y5Y4 3/20 0.39
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
IDH1 O75874 2/20 0.37
NPY5R Q15761 1/20 0.37
ALOX5 P09917 1/20 0.37
AKR1B1 P15121 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637173 0.86 AKR1C3 (0.45) AKR1C3SPRSRCAKR1C2KIF11
SCHEMBL28626501 0.86 SPR (0.44) AKR1C3SPRTACR1SRCAKR1C2
SCHEMBL28621882 0.84 SPR (0.51) AKR1C3SPRTACR1AKR1C2TSHR
SCHEMBL28621975 0.81 MEN1 (0.51) SRCKDM4EMAPTHPGDNPY5R
SCHEMBL28621885 0.79 MEN1 (0.51) SPRTACR1SRCPTGDR2KDM4E
SCHEMBL17968711 0.78 KIF11 (0.49) AKR1C3SPRSRCAKR1C2KIF11
SCHEMBL29160660 0.78 SPR (0.50) AKR1C3SPRAKR1C2TSHRKDM4E
SCHEMBL18015724 0.76 KIF11 (0.50) AKR1C3SRCAKR1C2KIF11CYP2C9
SCHEMBL28631063 0.75 MEN1 (0.50) SPRSRCAKR1C2KIF11KDM4E
SCHEMBL18014737 0.74 KIF11 (0.48) AKR1C3SRCAKR1C2KIF11CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429332-B 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2023-12-15 CN disclosed
CN-113429332-A 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2021-09-24 CN disclosed