SCHEMBL28637173

SCHEMBL28637173

Cc1c(CCC(=O)O)c2cc(C(F)(F)F)ccc2n1C

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.45
AKR1C2 P52895 5/20 0.45
PTGDR2 Q9Y5Y4 3/20 0.45
PLA2G4A P47712 1/20 0.45
PDE5A O76074 1/20 0.44
PDE9A O76083 1/20 0.44
EGFR P00533 1/20 0.43
SRC P12931 1/20 0.43
KMO O15229 1/20 0.43
KIF11 P52732 1/20 0.43
CYP2C9 P11712 1/20 0.42
SPR P35270 1/20 0.41
PTGS1 P23219 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
FFAR1 O14842 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28626909 0.86 AKR1C3 (0.47) AKR1C3AKR1C2PTGDR2SRCKIF11
SCHEMBL28626501 0.86 SPR (0.44) AKR1C3AKR1C2PTGDR2SRCKIF11
SCHEMBL20120108 0.82 KDM4E (0.50) AKR1C3AKR1C2PTGDR2PLA2G4AEGFR
SCHEMBL34461880 0.82 EGFR (0.47) PLA2G4AEGFRSPRNR1H4
SCHEMBL28621975 0.82 MEN1 (0.51) SRC
SCHEMBL18509545 0.81 SPR (0.59) AKR1C3AKR1C2PLA2G4AEGFRSPR
SCHEMBL17968711 0.81 KIF11 (0.49) AKR1C3AKR1C2PTGDR2EGFRSRC
SCHEMBL18509564 0.80 AKR1C3 (0.56) AKR1C3AKR1C2PLA2G4AEGFRKMO
SCHEMBL18509730 0.80 PLA2G4A (0.47) AKR1C3AKR1C2PLA2G4APDE5APDE9A
SCHEMBL18509742 0.80 PLA2G2A (0.48) AKR1C3AKR1C2PLA2G4AEGFRSPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429332-B 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2023-12-15 CN disclosed
CN-113429332-A 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2021-09-24 CN disclosed