SCHEMBL28627152

SCHEMBL28627152

CCC(=O)N(c1ccccc1)C1CCN(c2cc(C(F)(F)F)ccc2CN2CCN(C(=O)OC(C)(C)C)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 11/20 0.53
ABHD6 Q9BV23 9/20 0.53
PLA2G7 Q13093 5/20 0.53
OPRM1 P35372 2/20 0.51
CYP2D6 P10635 1/20 0.51
SIGMAR1 Q99720 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
FAAH O00519 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28613846 0.89 OPRM1 (0.55) MGLLABHD6PLA2G7OPRM1SIGMAR1
SCHEMBL28627150 0.88 OPRM1 (0.50) MGLLABHD6PLA2G7OPRM1CYP2D6
SCHEMBL30632159 0.86 OPRM1 (0.55) OPRM1SIGMAR1
SCHEMBL28612071 0.86 OPRM1 (0.55) OPRM1SIGMAR1
SCHEMBL28614771 0.85 OPRM1 (0.47) MGLLABHD6PLA2G7OPRM1CYP2D6
SCHEMBL30632157 0.85 OPRM1 (0.47) MGLLABHD6PLA2G7OPRM1CYP2D6
Tert-Butyl Formate SCHEMBL28627151 0.84 OPRM1 (0.48) MGLLABHD6PLA2G7OPRM1SIGMAR1
SCHEMBL30632156 0.84 MGLL (0.56) MGLLABHD6PLA2G7CYP2D6FAAH
SCHEMBL28614777 0.84 MGLL (0.56) MGLLABHD6PLA2G7CYP2D6FAAH
SCHEMBL20567165 0.81 MGLL (0.59) MGLLABHD6PLA2G7CYP2D6FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113292485-B Benzyl piperazine urea TRPV1 antagonizing and MOR agonizing double-target medicine and its prepn and application 河南大学 2023-10-27 CN disclosed
CN-113292485-A Benzylpiperazine urea TRPV1 antagonistic and MOR agonistic double-target-point medicine, preparation method and application 河南大学 2021-08-24 CN disclosed