SCHEMBL28627150

SCHEMBL28627150

CCC(=O)N(c1ccccc1)C1CCN(c2cc(C(F)(F)F)ccc2CN2CCN(OC(=O)C(C)(C)C)CC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.50
SIGMAR1 Q99720 2/20 0.48
MGLL Q99685 4/20 0.44
ABHD6 Q9BV23 4/20 0.44
PLA2G7 Q13093 3/20 0.44
OPRD1 P41143 2/20 0.43
SLC22A1 O15245 1/20 0.43
NR1I2 O75469 1/20 0.43
ABCB1 P08183 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
CHRM3 P20309 1/20 0.43
MAOA P21397 1/20 0.43
DRD4 P21917 1/20 0.43
MAOB P27338 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
ADRA1B P35368 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28612072 0.89 OPRM1 (0.54) OPRM1SIGMAR1OPRD1SLC22A1NR1I2
SCHEMBL28627152 0.88 MGLL (0.53) OPRM1SIGMAR1MGLLABHD6PLA2G7
SCHEMBL28612071 0.85 OPRM1 (0.55) OPRM1SIGMAR1OPRD1SLC22A1NR1I2
SCHEMBL30632159 0.85 OPRM1 (0.55) OPRM1SIGMAR1OPRD1SLC22A1NR1I2
Tert-Butyl Formate SCHEMBL28627151 0.82 OPRM1 (0.48) OPRM1SIGMAR1MGLLABHD6PLA2G7
SCHEMBL30632157 0.82 OPRM1 (0.47) OPRM1SIGMAR1MGLLABHD6PLA2G7
SCHEMBL28614771 0.82 OPRM1 (0.47) OPRM1SIGMAR1MGLLABHD6PLA2G7
SCHEMBL27994101 0.81 MGLL (0.61) MGLLABHD6PLA2G7CYP2D6
SCHEMBL28613846 0.76 OPRM1 (0.55) OPRM1SIGMAR1MGLLABHD6PLA2G7
SCHEMBL28620550 0.76 OPRM1 (0.58) OPRM1SIGMAR1OPRD1SLC22A1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113292485-A Benzylpiperazine urea TRPV1 antagonistic and MOR agonistic double-target-point medicine, preparation method and application 河南大学 2021-08-24 CN disclosed