SCHEMBL28629490

SCHEMBL28629490

CC(=O)OC(OC(N)=O)c1ccccc1.c1cc2ccc1-2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
MMP12 P39900 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TSHR P16473 1/20 0.40
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTGS2 P35354 1/20 0.40
MAPT P10636 1/20 0.39
ACP3 P15309 1/20 0.39
PABPC1 P11940 1/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
ALOX5 P09917 1/20 0.38
CYP19A1 P11511 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9939344 0.95 PTGS2 (0.46) ALDH1A1CYP3A4MMP12SMN1; SMN2CYP1A2
SCHEMBL27679472 0.95 ALDH1A1 (0.54) ALDH1A1CYP3A4SMN1; SMN2CYP1A2CYP2D6
SCHEMBL4198693 0.86 PTGS2 (0.53) ALDH1A1CYP3A4MMP12SMN1; SMN2CYP1A2
SCHEMBL5306707 0.86 CYP2D6 (0.52) ALDH1A1CYP3A4SMN1; SMN2CYP1A2CYP2D6
SCHEMBL486678 0.86 ALDH1A1 (0.63) ALDH1A1CYP3A4CYP2D6TSHRHSD17B10
SCHEMBL14798131 0.84 ALDH1A1 (0.61) ALDH1A1CYP3A4CYP2D6TSHRHSD17B10
SCHEMBL28881766 0.83 ALDH1A1 (0.50) ALDH1A1CYP3A4MMP12SMN1; SMN2CYP1A2
SCHEMBL113808 0.79 CYP2D6 (0.46) ALDH1A1CYP3A4SMN1; SMN2CYP1A2CYP2D6
SCHEMBL27601373 0.78 ALDH1A1 (0.51) ALDH1A1CYP3A4MMP12SMN1; SMN2TSHR
SCHEMBL6372424 0.77 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2D6TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113226377-B Antibody drug conjugates comprising an eltrinastine derivative 法马马有限公司 2022-10-18 CN disclosed
CN-113226377-A Antibody drug conjugates comprising an eltrinastine derivative 法马马有限公司 2021-08-06 CN disclosed