SCHEMBL28631402

SCHEMBL28631402

Cc1cccc(F)c1-c1cc2ccncc2cc1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 3/20 0.49
NCOA3 Q9Y6Q9 1/20 0.41
HTT P42858 1/20 0.40
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
HASPIN Q8TF76 1/20 0.40
CYP11B1 P15538 3/20 0.37
CYP11B2 P19099 3/20 0.37
DYRK1A Q13627 6/20 0.35
CLK1 P49759 5/20 0.35
CLK2 P49760 5/20 0.35
CLK4 Q9HAZ1 5/20 0.35
DYRK1B Q9Y463 4/20 0.35
CDK5 Q00535 4/20 0.35
CDK5R1 Q15078 4/20 0.35
CLK3 P49761 3/20 0.35
PIM2 Q9P1W9 1/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930315 1.00 MAP4K1 (0.49) MAP4K1NCOA3HTTCCNT1CDK9
SCHEMBL28925081 0.78 MAP4K1 (0.43) MAP4K1DYRK1AALDH1A1
SCHEMBL28635707 0.77 MAP4K1 (0.43) MAP4K1NCOA3CYP11B2ALDH1A1
SCHEMBL28634082 0.76 MAP4K1 (0.43) MAP4K1ALDH1A1KDM4EGAA
SCHEMBL18050177 0.75 CCNT1 (0.53) NCOA3HTTCCNT1CDK9HASPIN
SCHEMBL23301805 0.69 F7 (0.38) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL29897403 0.69 F7 (0.38) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL28633555 0.69 MAP4K1 (0.42) MAP4K1HTTCYP11B1CYP11B2
SCHEMBL23962778 0.68 MAP4K1 (0.41) MAP4K1GAA
SCHEMBL28284386 0.68 MAP4K1 (0.38) MAP4K1CYP11B1CYP11B2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115244050-B Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2024-06-21 CN disclosed
CN-115244050-A Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2022-10-25 CN disclosed
CN-113336747-A Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2021-09-03 CN disclosed