SCHEMBL28635707

SCHEMBL28635707

Cc1cccc(F)c1-c1cc2ccnc(Cl)c2cc1C#N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 2/20 0.43
ALDH1A1 P00352 1/20 0.41
KHK P50053 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
EGLN2 Q96KS0 3/20 0.33
CYP11B2 P19099 1/20 0.33
TGFBR1 P36897 1/20 0.32
TYK2 P29597 1/20 0.32
KDM1A O60341 2/20 0.32
LRRK2 Q5S007 1/20 0.32
USP8 P40818 1/20 0.32
MAPK14 Q16539 1/20 0.31
ORAI1 Q96D31 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28925081 0.87 MAP4K1 (0.43) MAP4K1ALDH1A1KHKEGLN2KDM1A
SCHEMBL28631402 0.77 MAP4K1 (0.49) MAP4K1ALDH1A1CYP11B2NCOA3
SCHEMBL29930315 0.77 MAP4K1 (0.49) MAP4K1ALDH1A1CYP11B2NCOA3
SCHEMBL28631850 0.75 WNT3A (0.43) ALDH1A1TYK2MAPK14
SCHEMBL29929742 0.75 WNT3A (0.43) ALDH1A1TYK2MAPK14
SCHEMBL16858473 0.74 KHK (0.42) ALDH1A1KHKNPSR1EGLN2CYP11B2
SCHEMBL28551219 0.74 ALDH1A1 (0.46) ALDH1A1KHKCYP1A2CYP2C9CYP2C19
SCHEMBL28633555 0.71 MAP4K1 (0.42) MAP4K1EGLN2CYP11B2KDM1A
SCHEMBL15820110 0.71 ALDH1A1 (0.40) MAP4K1ALDH1A1KHKNPSR1LRRK2
SCHEMBL15428069 0.69 PARG (0.37) CYP1A2CYP2C9CYP2C19SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115244050-B Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2024-06-21 CN disclosed
CN-115244050-A Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2022-10-25 CN disclosed
CN-113336747-A Novel HPK1 inhibitor and preparation method and application thereof 轶诺(浙江)药业有限公司 2021-09-03 CN disclosed