SCHEMBL28633205

SCHEMBL28633205

Cn1ccc(-c2ccc(NC(=O)O)cc2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
KEAP1 Q14145 1/20 0.51
NPC1 O15118 5/20 0.47
KDM4E B2RXH2 5/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
RAB9A P51151 5/20 0.45
IKBKE Q14164 1/20 0.45
TBK1 Q9UHD2 1/20 0.45
CREBBP Q92793 2/20 0.44
BRD4 O60885 1/20 0.44
SCN4A P35499 1/20 0.44
MAPT P10636 3/20 0.44
PKM P14618 1/20 0.44
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP19A1 P11511 1/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14069326 0.83 TSHR (0.50) KMT2AKEAP1NPC1IKBKETBK1
SCHEMBL29796107 0.81 KMT2A (0.53) KMT2ANPC1KDM4ESMN1; SMN2RAB9A
SCHEMBL31323274 0.80 TAAR1 (0.57) KMT2AKEAP1NPC1KDM4ESMN1; SMN2
SCHEMBL31306170 0.80 MAPT (0.47) KMT2AKEAP1NPC1KDM4ESMN1; SMN2
SCHEMBL31306229 0.80 KEAP1 (0.45) KMT2AKEAP1NPC1KDM4ESMN1; SMN2
SCHEMBL31323277 0.80 TAAR1 (0.57) KMT2AKEAP1NPC1KDM4ESMN1; SMN2
SCHEMBL21286259 0.80 KMT2A (0.60) KMT2ANPC1KDM4ESMN1; SMN2RAB9A
SCHEMBL14199838 0.79 RAB9A (0.56) KMT2ANPC1KDM4ESMN1; SMN2RAB9A
SCHEMBL2629322 0.77 KMT2A (0.60) KMT2AKEAP1NPC1KDM4ESMN1; SMN2
SCHEMBL28937613 0.77 KEAP1 (0.60) KMT2AKEAP1NPC1IKBKETBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed