SCHEMBL28633762

SCHEMBL28633762

[CH2]C(=O)NNC(=S)Nc1ccc(Br)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.66
PKM P14618 1/20 0.66
MEN1 O00255 5/20 0.62
KMT2A Q03164 5/20 0.62
RAB9A P51151 1/20 0.62
ALDH1A1 P00352 5/20 0.59
MAPT P10636 4/20 0.59
EPHX1 P07099 2/20 0.57
MAOA P21397 2/20 0.55
MAOB P27338 2/20 0.55
IDO1 P14902 1/20 0.55
LMNA P02545 3/20 0.53
HTT P42858 2/20 0.53
MAPK1 P28482 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
KDM4E B2RXH2 1/20 0.51
F13A1 P00488 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633748 0.82 NOX1 (0.66) GAAPKMMEN1KMT2ARAB9A
SCHEMBL28641155 0.82 NOX1 (0.66) GAAPKMMEN1KMT2ARAB9A
SCHEMBL28651984 0.82 ALDH1A1 (0.64) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL28636321 0.81 GAA (0.73) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL28641144 0.80 ALDH1A1 (0.61) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL25132398 0.78 GAA (0.60) GAAPKMMEN1KMT2ARAB9A
SCHEMBL28924353 0.78 EPHX2 (0.56) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL28640790 0.78 GAA (0.61) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL5455602 0.78 MAPT (0.83) GAAMEN1KMT2ARAB9AALDH1A1
SCHEMBL8956372 0.78 MAPT (0.83) GAAMEN1KMT2ARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113480524-A Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2021-10-08 CN claimed
CN-113480524-B Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2022-08-30 CN disclosed
CN-113480524-A Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2021-10-08 CN disclosed