SCHEMBL28634875

SCHEMBL28634875

CC(C)(C)OC(=O)N1CCN(Cc2nc3ccc(Br)cc3c(=O)[nH]2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
LMNA P02545 1/20 0.50
GAA P10253 4/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
ALDH1A1 P00352 4/20 0.46
PIM1 P11309 4/20 0.46
CSNK2A2 P19784 4/20 0.46
CSNK2B P67870 4/20 0.46
PIM3 Q86V86 4/20 0.46
PIM2 Q9P1W9 4/20 0.46
POLB P06746 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
IDO2 Q6ZQW0 1/20 0.46
DRD4 P21917 2/20 0.45
CDC7 O00311 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29111354 0.86 GAA (0.66) LMNAGAAL3MBTL1ALDH1A1POLB
SCHEMBL31569732 0.85 TBK1 (0.44) MAPTLMNADRD4
SCHEMBL30669819 0.84 GAA (0.55) MAPTLMNAGAAL3MBTL1ALDH1A1
SCHEMBL28627494 0.84 GAA (0.55) MAPTLMNAGAAL3MBTL1ALDH1A1
SCHEMBL26170030 0.83 NAMPT (0.51)
SCHEMBL23293923 0.79 KDM4E (0.47) MAPTALDH1A1HPGDNPSR1
SCHEMBL30947729 0.79 KDM4E (0.47) MAPTALDH1A1HPGDNPSR1
SCHEMBL30186938 0.79 NSD2 (0.47) MAPTL3MBTL1ALDH1A1PIM1PIM2
SCHEMBL26170074 0.79 NSD2 (0.47) MAPTL3MBTL1ALDH1A1PIM1PIM2
SCHEMBL30947756 0.78 JAK2 (0.40) MAPTGAAIDO1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461661-B 6- (pyridin-3-yl) quinazoline-4 (3H) -ketone derivative and preparation and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2023-11-28 CN disclosed
CN-113461661-A 6- (pyridine-3-yl) quinazoline-4 (3H) -ketone derivative and preparation and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2021-10-01 CN disclosed