SCHEMBL28635157

SCHEMBL28635157

COc1ccc(Nc2ncnc3cc(OCCCCl)c(OC)cc23)cc1OC

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.79
CLK1 P49759 2/20 0.79
ABCG2 Q9UNQ0 1/20 0.79
LCK P06239 2/20 0.77
KDR P35968 5/20 0.65
RET P07949 2/20 0.65
KIF5B P33176 2/20 0.65
FLT1 P17948 1/20 0.65
SRC P12931 1/20 0.63
AURKA O14965 1/20 0.61
ERBB2 P04626 1/20 0.61
INSR P06213 1/20 0.61
FBP1 P09467 1/20 0.61
PDGFRB P09619 1/20 0.61
FLT4 P35916 1/20 0.61
EPHB4 P54760 1/20 0.61
TEK Q02763 1/20 0.61
AURKB Q96GD4 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28646400 0.90 KDR (0.80) EGFRABCG2LCKKDRRET
SCHEMBL5565137 0.89 EGFR (1.00) EGFRCLK1ABCG2LCKKDR
SCHEMBL14964688 0.89 EGFR (0.80) EGFRLCKKDRFLT1
SCHEMBL14964773 0.87 EGFR (0.85) EGFRCLK1KDRAURKAERBB2
SCHEMBL31491085 0.87 EGFR (0.85) EGFRCLK1KDRAURKAERBB2
SCHEMBL30207668 0.87 EGFR (0.85) EGFRCLK1KDRAURKAERBB2
SCHEMBL28520911 0.87 EGFR (0.85) EGFRCLK1KDRAURKAERBB2
SCHEMBL28641557 0.86 FBP1 (0.83) EGFRABCG2KDRFLT1SRC
SCHEMBL6691545 0.85 KDR (0.60) EGFRCLK1ABCG2LCKKDR
SCHEMBL6691540 0.85 KDR (0.66) EGFRKDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106083836-B H based on quinazoline structure2S donor compound and application thereof 徐州医学院 2021-08-20 CN disclosed