SCHEMBL28635648

SCHEMBL28635648

O=C(O)c1nc2cnccc2n1C1CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 3/20 0.48
CYP2D6 P10635 1/20 0.45
CCR5 P51681 1/20 0.45
CYP11B2 P19099 4/20 0.44
CYP11B1 P15538 2/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OGFRL1 Q5TC84 1/20 0.39
ATM Q13315 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4D Q08499 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP3A4 P08684 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23624207 0.83 RPS6KA5 (0.44) RPS6KA5CYP2D6CCR5CYP11B2CYP11B1
SCHEMBL16083674 0.75 RPS6KA5 (0.52) RPS6KA5CYP2D6CCR5CYP11B2CYP11B1
SCHEMBL927948 0.75 CYP1A2 (0.64) RPS6KA5CYP2D6CYP11B2ATMCYP3A4
SCHEMBL4138903 0.73 CCR5 (0.58) RPS6KA5CYP2D6CCR5L3MBTL1ALDH1A1
SCHEMBL30497300 0.72 PDE4B (0.52) OPRM1OPRD1OPRK1OGFRL1PDE4B
SCHEMBL28645924 0.72 RPS6KA5 (0.49) RPS6KA5CYP2D6ATMALDH1A1CYP2C19
SCHEMBL3064217 0.70 CCR5 (0.47) RPS6KA5CYP2D6CCR5CYP11B2L3MBTL1
SCHEMBL3064218 0.70 CCR5 (0.47) RPS6KA5CYP2D6CCR5CYP11B2L3MBTL1
SCHEMBL19851139 0.69 RPS6KA5 (0.55) RPS6KA5CYP2D6CCR5CYP11B2CYP11B1
SCHEMBL16054503 0.69 RPS6KA5 (0.55) RPS6KA5CYP2D6CCR5CYP11B2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113348170-B Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-22 CN disclosed
CN-113348170-A Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-03 CN disclosed