SCHEMBL28645924

SCHEMBL28645924

CCn1c(C(=O)O)nc2cnccc21

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 8/20 0.49
RPS6KB1 P23443 1/20 0.47
CDK2 P24941 1/20 0.47
ROCK1 Q13464 1/20 0.47
DYRK1A Q13627 1/20 0.47
RPS6KA1 Q15418 1/20 0.47
S1PR1 P21453 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM5A P29375 1/20 0.42
PTGER4 P35408 2/20 0.41
SLC22A12 Q96S37 1/20 0.41
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ATM Q13315 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23624032 0.84 RPS6KA5 (0.49) RPS6KA5RPS6KB1CDK2ROCK1DYRK1A
SCHEMBL3619365 0.80 MAPK1 (0.61) CYP2D6MAPK1CASP1CASP7ALDH1A1
SCHEMBL13071643 0.78 RPS6KA5 (0.54) RPS6KA5RPS6KB1CDK2ROCK1DYRK1A
SCHEMBL4717496 0.72 TP53 (0.47) RPS6KA5RPS6KB1CDK2ROCK1DYRK1A
SCHEMBL28635648 0.72 RPS6KA5 (0.48) RPS6KA5CYP2D6CYP2C19SLC22A12ATM
SCHEMBL8322125 0.71 L3MBTL1 (0.46) RPS6KA5ATM
SCHEMBL12085751 0.70 GPR35 (0.55) KDM5APTGER4ALDH1A1
SCHEMBL13497676 0.70 S1PR1 (0.54) RPS6KA5RPS6KB1CDK2ROCK1DYRK1A
SCHEMBL7496365 0.70
SCHEMBL7501624 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113348170-B Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-22 CN disclosed
CN-113348170-A Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-03 CN disclosed