SCHEMBL28635974

SCHEMBL28635974

CC(C)(C)OC(=O)n1c(=O)n(C(=O)O)c2cc(Br)ccc21

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
CCNB2 O95067 1/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
GSK3B P49841 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43
USP30 Q70CQ3 2/20 0.37
NR1H2 P55055 9/20 0.37
NR1H3 Q13133 2/20 0.37
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
MCL1 Q07820 1/20 0.35
RORC P51449 2/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16262449 0.94 ALDH1A1 (0.48) ALDH1A1CCNB2CDK1CCNB1GSK3B
SCHEMBL31710152 0.85 LMNA (0.48) ALDH1A1CCNB2CDK1CCNB1GSK3B
SCHEMBL5418830 0.85 CCNB2 (0.44) ALDH1A1CCNB2CDK1CCNB1GSK3B
SCHEMBL31709563 0.78 ALDH1A1 (0.45) ALDH1A1CCNB2CDK1CCNB1GSK3B
SCHEMBL409607 0.77 CDK1 (0.54) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL31709387 0.76 ALDH1A1 (0.43) ALDH1A1CCNB2CDK1CCNB1GSK3B
SCHEMBL31709866 0.76 AKT2 (0.44) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL7479161 0.75 MCL1 (0.47) ALDH1A1MCL1
SCHEMBL13429972 0.74 CCNB2 (0.42) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL8222044 0.73 LMNA (0.39) NR1H2NR1H3GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113543783-A Kinase inhibitor compounds and compositions and methods of use 西奈山伊坎医学院 2021-10-22 CN disclosed
CN-113508111-A Kinase inhibitor compounds and compositions and methods of use 西奈山伊坎医学院 2021-10-15 CN disclosed