SCHEMBL28636737

SCHEMBL28636737

O=C(OCBr)c1ccc(CBr)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 2/20 0.53
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 3/20 0.44
ESR1 P03372 3/20 0.44
SLC6A2 P23975 2/20 0.44
ESR2 Q92731 2/20 0.44
SLC6A3 Q01959 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
MAPT P10636 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28716126 0.89 ESR1 (0.52) KMT2AMEN1LMNATDP1ESR1
SCHEMBL245250 0.86 CA1 (0.63) KMT2AMEN1LMNATDP1ESR1
SCHEMBL636176 0.84 CES2 (0.55) KMT2AMEN1CES2CES1LMNA
SCHEMBL2500365 0.84 CES2 (0.55) KMT2AMEN1CES2CES1LMNA
SCHEMBL8838298 0.84 TDP1 (0.58) KMT2AMEN1CES2CES1LMNA
SCHEMBL8617188 0.83 ALDH1A1 (0.66) KMT2AMEN1LMNATDP1ESR1
SCHEMBL28268071 0.83 CES2 (0.46) KMT2AMEN1CES2CES1LMNA
SCHEMBL8159484 0.83 CES2 (0.53) KMT2AMEN1CES2CES1LMNA
SCHEMBL7455670 0.81 ALDH1A1 (0.51) KMT2AMEN1CES2CES1ALDH1A1
SCHEMBL3158166 0.81 KMT2A (0.44) KMT2AMEN1CES2CES1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108341814-B JAK kinase inhibitors and uses thereof 上海翔锦生物科技有限公司 2021-09-03 CN disclosed