SCHEMBL28637102

SCHEMBL28637102

O=c1c(NCc2ccccn2)c(Nc2ccccc2)c1=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.63
MAOB P27338 3/20 0.63
MAPKAPK2 P49137 1/20 0.58
KCNH2 Q12809 2/20 0.51
CHEK1 O14757 3/20 0.50
CHEK2 O96017 3/20 0.50
PRKACA P17612 3/20 0.50
RPS6KB1 P23443 3/20 0.50
GSK3A P49840 3/20 0.50
GSK3B P49841 3/20 0.50
RPS6KA3 P51812 3/20 0.50
PRKCD Q05655 3/20 0.50
ROCK1 Q13464 3/20 0.50
PRKG1 Q13976 3/20 0.50
PKN2 Q16513 3/20 0.50
CDC42BPA Q5VT25 3/20 0.50
HIPK4 Q8NE63 3/20 0.50
AURKB Q96GD4 3/20 0.50
MKNK2 Q9HBH9 3/20 0.50
SGK2 Q9HBY8 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366437 0.91 MAPKAPK2 (0.68) MAOAMAOBMAPKAPK2KCNH2CHEK1
SCHEMBL28642296 0.89 CHEK2 (0.58) MAOAMAOBMAPKAPK2KCNH2CHEK1
SCHEMBL28925293 0.89 MAPKAPK2 (0.50) MAOAMAOBMAPKAPK2KCNH2CHEK1
SCHEMBL28651333 0.89 CHEK1 (0.52) MAOAMAOBMAPKAPK2CHEK1CHEK2
SCHEMBL28635668 0.89 MAPKAPK2 (0.50) MAOAMAOBMAPKAPK2KCNH2CHEK1
SCHEMBL28640083 0.89 KMT2A (0.53) MAOAMAOBMAPKAPK2KCNH2CHEK1
SCHEMBL28633070 0.89 CHEK1 (0.58) MAOAMAOBMAPKAPK2CHEK1CHEK2
SCHEMBL30513615 0.86 PIK3CA (0.51) MAOAMAOBMAPKAPK2KCNH2NPC1
SCHEMBL28637301 0.86 ABCB1 (0.57) MAOAMAOBMAPKAPK2CHEK1CHEK2
SCHEMBL28653147 0.86 PIK3CA (0.51) MAOAMAOBMAPKAPK2KCNH2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed
CN-112759549-A 3-substituted amino-4- ((substituted pyridyl) amino) cyclobut-3-ene-1, 2-diones 中国医学科学院药物研究所 2021-05-07 CN disclosed