SCHEMBL28635668

SCHEMBL28635668

O=c1c(NCc2ccccn2)c(Nc2ccc(O)cc2)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.50
MAOA P21397 3/20 0.49
MAOB P27338 3/20 0.49
CHEK1 O14757 3/20 0.46
CHEK2 O96017 3/20 0.46
PRKACA P17612 3/20 0.46
RPS6KB1 P23443 3/20 0.46
GSK3A P49840 3/20 0.46
GSK3B P49841 3/20 0.46
RPS6KA3 P51812 3/20 0.46
PRKCD Q05655 3/20 0.46
ROCK1 Q13464 3/20 0.46
PRKG1 Q13976 3/20 0.46
PKN2 Q16513 3/20 0.46
CDC42BPA Q5VT25 3/20 0.46
HIPK4 Q8NE63 3/20 0.46
AURKB Q96GD4 3/20 0.46
MKNK2 Q9HBH9 3/20 0.46
SGK2 Q9HBY8 3/20 0.46
CSNK1G3 Q9Y6M4 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637102 0.89 MAOA (0.63) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL30513615 0.87 PIK3CA (0.51) MAPKAPK2MAOAMAOBSMN1; SMN2ALDH1A1
SCHEMBL28653147 0.87 PIK3CA (0.51) MAPKAPK2MAOAMAOBSMN1; SMN2ALDH1A1
SCHEMBL28640083 0.86 KMT2A (0.53) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL28925293 0.86 MAPKAPK2 (0.50) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL28651333 0.86 CHEK1 (0.52) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL28642296 0.86 CHEK2 (0.58) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL28633070 0.86 CHEK1 (0.58) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL4366437 0.86 MAPKAPK2 (0.68) MAPKAPK2MAOAMAOBCHEK1CHEK2
SCHEMBL28637146 0.85 SMN1; SMN2 (0.49) MAPKAPK2MAOAMAOBCHEK1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed
CN-112759549-A 3-substituted amino-4- ((substituted pyridyl) amino) cyclobut-3-ene-1, 2-diones 中国医学科学院药物研究所 2021-05-07 CN disclosed