SCHEMBL28653147

SCHEMBL28653147

O=c1c(NCc2ccccn2)c(Nc2cccc(O)c2)c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.51
MTOR P42345 1/20 0.51
MAOA P21397 2/20 0.50
MAOB P27338 2/20 0.50
ITGB3 P05106 1/20 0.49
ITGAV P06756 1/20 0.49
SMN1; SMN2 Q16637 5/20 0.47
ALOX15 P16050 1/20 0.47
MAPKAPK2 P49137 1/20 0.45
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
STAT3 P40763 1/20 0.44
STAT1 P42224 1/20 0.44
TSHR P16473 2/20 0.43
CYP3A4 P08684 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KCNH2 Q12809 1/20 0.43
KMT2A Q03164 1/20 0.43
MBD2 Q9UBB5 1/20 0.43
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30513615 1.00 PIK3CA (0.51) PIK3CAMTORMAOAMAOBITGB3
SCHEMBL28635668 0.87 MAPKAPK2 (0.50) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL28637102 0.86 MAOA (0.63) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL30513603 0.86 KMT2A (0.56) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL28637137 0.86 KMT2A (0.56) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL28652875 0.84 GRM4 (0.48) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL30513604 0.84 GRM4 (0.48) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL30513599 0.83 KMT2A (0.63) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL28641996 0.83 KMT2A (0.63) MAOAMAOBITGB3ITGAVSMN1; SMN2
SCHEMBL4366437 0.81 MAPKAPK2 (0.68) MAOAMAOBMAPKAPK2CYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed
CN-112759549-A 3-substituted amino-4- ((substituted pyridyl) amino) cyclobut-3-ene-1, 2-diones 中国医学科学院药物研究所 2021-05-07 CN disclosed