SCHEMBL4366437

SCHEMBL4366437

O=c1c(NCc2ccccn2)c(Nc2ccncc2)c1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 6/20 0.68
ROCK1 Q13464 9/20 0.61
AURKB Q96GD4 9/20 0.61
GSK3A P49840 8/20 0.61
GSK3B P49841 8/20 0.61
CDC42BPA Q5VT25 8/20 0.61
CSNK1G3 Q9Y6M4 8/20 0.61
PRKACA P17612 7/20 0.61
RPS6KB1 P23443 7/20 0.61
RPS6KA3 P51812 7/20 0.61
CHEK2 O96017 7/20 0.61
PRKG1 Q13976 6/20 0.61
PKN2 Q16513 6/20 0.61
HIPK4 Q8NE63 6/20 0.61
CHEK1 O14757 5/20 0.61
MKNK2 Q9HBH9 5/20 0.61
SGK2 Q9HBY8 5/20 0.61
AKT1 P31749 5/20 0.61
PRKCD Q05655 4/20 0.61
PRKAA1 Q13131 4/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637102 0.91 MAOA (0.63) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28633070 0.86 CHEK1 (0.58) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28635668 0.86 MAPKAPK2 (0.50) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28651333 0.86 CHEK1 (0.52) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28925293 0.86 MAPKAPK2 (0.50) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28640083 0.86 KMT2A (0.53) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28642296 0.86 CHEK2 (0.58) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28637301 0.84 ABCB1 (0.57) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL28651862 0.83 NPC1 (0.54) MAPKAPK2ROCK1AURKBGSK3AGSK3B
SCHEMBL30513612 0.83 MAOA (0.69) MAPKAPK2ROCK1AURKBGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO claimed
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed