SCHEMBL28637205

SCHEMBL28637205

Nc1c(C(=O)O)ccc(-c2ccccc2)c1-c1cnc[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
MEN1 O00255 2/20 0.49
THRB P10828 2/20 0.49
MAPK1 P28482 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.49
RECQL P46063 1/20 0.49
IDO1 P14902 7/20 0.47
CYP3A4 P08684 2/20 0.47
FTO Q9C0B1 1/20 0.46
HPGDS O60760 1/20 0.41
KDM4E B2RXH2 1/20 0.39
USP2 O75604 1/20 0.39
PKM P14618 1/20 0.39
MCL1 Q07820 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
FNTA P49354 2/20 0.39
FNTB P49356 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2462914 0.78 MEN1 (0.60) MAPTMEN1THRBMAPK1KMT2A
SCHEMBL28640384 0.77 FTO (0.38) IDO1CYP3A4FTOHPGDSFNTA
SCHEMBL21857697 0.74 IDO1 (0.54) MAPTMEN1THRBMAPK1KMT2A
SCHEMBL28636872 0.73 FTO (0.44) KMT2AALDH1A1IDO1CYP3A4FTO
SCHEMBL28926573 0.73 FTO (0.44) KMT2AALDH1A1IDO1CYP3A4FTO
SCHEMBL980179 0.73 IDO1 (0.46) MAPK1IDO1CYP3A4HPGDSCSF1R
SCHEMBL6316181 0.71 ALDH1A1 (0.54) MAPTMEN1THRBMAPK1KMT2A
SCHEMBL2417930 0.69 IDO1 (0.45) IDO1CYP3A4HPGDSCSF1RCYP2E1
SCHEMBL4849742 0.69 ALDH1A1 (0.51) MAPTMEN1THRBMAPK1KMT2A
SCHEMBL21857476 0.68 KMT2A (0.59) MAPTMEN1THRBKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed