SCHEMBL28640384

SCHEMBL28640384

NC(=O)c1c(C(=O)O)c(O)cc(C(=O)O)c1-c1c(C(=O)O)ccc(-c2ccccc2)c1-c1cnc[nH]1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 1/20 0.38
IDO1 P14902 8/20 0.38
CYP3A4 P08684 1/20 0.37
CSF1R P07333 2/20 0.36
PARP1 P09874 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
HPGDS O60760 1/20 0.33
MKNK1 Q9BUB5 2/20 0.33
MKNK2 Q9HBH9 2/20 0.33
CDC7 O00311 1/20 0.33
HNF4A P41235 2/20 0.33
ACMSD Q8TDX5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637205 0.77 MAPT (0.49) FTOIDO1CYP3A4CSF1RFNTA
SCHEMBL28636872 0.73 FTO (0.44) FTOIDO1CYP3A4CSF1RFNTA
SCHEMBL28926573 0.73 FTO (0.44) FTOIDO1CYP3A4CSF1RFNTA
SCHEMBL21857697 0.65 IDO1 (0.54) FTOIDO1CYP3A4PARP1HPGDS
Benzene SCHEMBL27914219 0.64 BCAT2 (0.50) MKNK1HNF4AACMSD
SCHEMBL28475228 0.64 BCAT2 (0.50) MKNK1HNF4AACMSD
SCHEMBL27639675 0.64 BCAT2 (0.50) MKNK1HNF4AACMSD
SCHEMBL28353064 0.64 BCAT2 (0.50) MKNK1HNF4AACMSD
SCHEMBL27323238 0.64 IDO1 (0.59) FTOIDO1CYP3A4PARP1
SCHEMBL2417930 0.63 IDO1 (0.45) IDO1CYP3A4CSF1RHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed