SCHEMBL28638604

SCHEMBL28638604

O=C(O)C(=O)Cc1ccc(F)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.55
CA2 P00918 1/20 0.47
RPA1 P27694 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
CNR2 P34972 1/20 0.44
F2 P00734 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
PLG P00747 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
C1S P09871 1/20 0.42
PRSS3 P35030 1/20 0.42
HAO1 Q9UJM8 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL869116 0.85 CA2 (0.65) PIK3CACA2RPA1ALDH1A1HDAC3
SCHEMBL2791406 0.84 PIK3CA (0.54) PIK3CACA2RPA1CNR2HDAC3
SCHEMBL9508267 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP3A4CYP2C19F2
SCHEMBL2164422 0.83 HAO1 (0.57) PIK3CACA2ALDH1A1CYP1A2CYP3A4
SCHEMBL21090110 0.81 PIK3CA (0.58) PIK3CACA2RPA1ALDH1A1CNR2
SCHEMBL28638605 0.80 PIK3CA (0.50) PIK3CACA2RPA1CNR2HDAC3
SCHEMBL11520973 0.80 PIK3CA (0.56) PIK3CACA2RPA1ALDH1A1CNR2
SCHEMBL3396522 0.80 PIK3CA (0.56) PIK3CACA2RPA1HDAC3HDAC1
SCHEMBL1699595 0.80 PIK3CA (0.56) PIK3CACA2RPA1ALDH1A1CNR2
SCHEMBL27835202 0.80 PIK3CA (0.56) PIK3CACA2RPA1ALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109761986-B Tricyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-10-08 CN disclosed