SCHEMBL2864153

SCHEMBL2864153

COc1ncc(CCN)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.47
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
HTR2B P41595 2/20 0.44
MAOB P27338 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
TSHR P16473 2/20 0.40
MAPK1 P28482 1/20 0.40
LMNA P02545 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
NFKB1 P19838 1/20 0.39
GLA P06280 1/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2760680 0.82 LOXL2 (0.44) TAAR1MAOBTUBB4ATUBBTUBA3C
Hydrochloric Acid SCHEMBL18130127 0.80 LOXL2 (0.42) MAOBTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL19219145 0.79 TUBB4A (0.36) HTR2ATUBB4ATUBBTUBA3CTUBA1B
SCHEMBL26393934 0.75 CASP3 (0.51) HTR2AHTR2CKDM4EATMTSHR
SCHEMBL19219147 0.75 TLR7 (0.36) TSHRCYP1A2CYP3A4TUBB4ATUBB
SCHEMBL7980765 0.75 CHRM2 (0.39) KDM4EGLATUBB4ATUBBTUBA3C
SCHEMBL20520312 0.75 GRM2 (0.41) LMNA
SCHEMBL8008816 0.75 TUBB4A (0.41) KDM4ETUBB4ATUBBTUBA3CTUBA1B
SCHEMBL2172820 0.75 TAAR1 (0.46) TAAR1HTR2AKDM4ECYP1A2CYP2A6
SCHEMBL23816857 0.74 CASP3 (0.50) HTR2AHTR2CKDM4EATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139334-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-01-06 EP disclosed
WO-2008130481-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-30 WO disclosed