SCHEMBL28643148

SCHEMBL28643148

O=C(O)c1nn2c(c1Br)CCCC2

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
TSHR P16473 1/20 0.31
GAA P10253 1/20 0.31
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28480405 0.95
SCHEMBL26978255 0.81 KMT2A (0.33) KMT2AHCAR2TSHRGAAALDH1A1
SCHEMBL31736856 0.78 CXCR4 (0.32)
SCHEMBL3801455 0.77 ALDH1A1 (0.40) KMT2ATSHRGAAALDH1A1POLB
SCHEMBL6382528 0.74 ALDH1A1 (0.34) KMT2AALDH1A1POLBMAPTL3MBTL1
SCHEMBL29777610 0.74 KDM4E (0.35) KMT2AALDH1A1POLBMAPTTDP1
SCHEMBL6384570 0.73 ALDH1A1 (0.36) ALDH1A1POLBMAPT
SCHEMBL29852457 0.73 ALDH1A1 (0.44) KMT2AGAAALDH1A1POLBMAPT
SCHEMBL31336737 0.72 GABRA1 (0.35) KMT2A
SCHEMBL6382734 0.69 GAA (0.33) KMT2AGAAALDH1A1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715632-B Macrocyclic indole derivatives 拜尔公开股份有限公司 2021-10-26 CN disclosed