SCHEMBL28645344

SCHEMBL28645344

CCOc1cc2c(cc1C(=O)O)CN(CC(C)(C)C)C2=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 1/20 0.41
LRRK2 Q5S007 2/20 0.37
ALOX15 P16050 1/20 0.37
CYP3A4 P08684 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.33
ACHE P22303 1/20 0.33
RXRA P19793 1/20 0.33
HNF4A P41235 1/20 0.33
TP53 P04637 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28926168 0.88 MEN1 (0.39) KMT2ATSHRHSD17B10LRRK2KDM4E
SCHEMBL28643695 0.85 LRRK2 (0.37) TSHRHSD17B10LRRK2ALOX15KDM4E
SCHEMBL28645763 0.83 KMT2A (0.41) KMT2ATSHRHSD17B10ALOX15
SCHEMBL28633462 0.81 KMT2A (0.53) KMT2AALOX15TP53
SCHEMBL28652352 0.80 KMT2A (0.48) KMT2ATSHRALOX15KDM4ETP53
SCHEMBL30604612 0.79 KMT2A (0.47) KMT2ATSHRCYP3A4LMNA
SCHEMBL28656930 0.79 KMT2A (0.45) KMT2ATSHRHSD17B10ALOX15TP53
SCHEMBL30604606 0.79 KMT2A (0.45) KMT2ATSHRHSD17B10ALOX15TP53
SCHEMBL28638917 0.79 KMT2A (0.47) KMT2ATSHRCYP3A4LMNA
SCHEMBL28644853 0.76 LRRK2 (0.42) KMT2ATSHRLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed