SCHEMBL28645446

SCHEMBL28645446

O=C(/C=C/c1cccc(O)c1)Nc1nncs1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.61
RAB9A P51151 4/20 0.61
KDM4E B2RXH2 2/20 0.61
ALDH1A1 P00352 1/20 0.61
MAPT P10636 1/20 0.61
SMN1; SMN2 Q16637 2/20 0.59
LMNA P02545 1/20 0.59
NFKB1 P19838 1/20 0.59
NFKB2 Q00653 1/20 0.59
RELA Q04206 1/20 0.59
MMP1 P03956 14/20 0.59
MMP2 P08253 14/20 0.59
MMP9 P14780 14/20 0.59
MAOB P27338 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31188414 1.00 NPC1 (0.61) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL6380999 0.85 RAB9A (0.70) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL6380992 0.85 RAB9A (0.70) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL13212214 0.83 AKT1 (0.58) MAPTMMP1MMP2MMP9MAOB
SCHEMBL28653222 0.80 NPC1 (0.76) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL31188413 0.80 NPC1 (0.76) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL22441647 0.75 LMNA (0.60) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL22441645 0.75 LMNA (0.60) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL28316655 0.75 MMP1 (1.00) MMP1MMP2MMP9MAOB
SCHEMBL14757343 0.74 NPC1 (1.00) NPC1RAB9AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603657-A Thiazolyl-containing propenone derivative and application thereof in preparation of kinase inhibitor 北京工业大学 2021-11-05 CN disclosed