SCHEMBL28645557

SCHEMBL28645557

[N-]=[N+]=NCc1cccc2c1ncn2CC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.46
CYP1A2 P05177 1/20 0.46
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
AR P10275 1/20 0.31
KAT2B Q92831 1/20 0.30
FDPS P14324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28636601 0.80 CYP17A1 (0.31) CYP17A1CYP1A2ARKAT2BFDPS
SCHEMBL21555726 0.78 CYP17A1 (0.54) CYP17A1CYP1A2ADORA2AADORA1AR
SCHEMBL28625938 0.78 CYP17A1 (0.51) CYP17A1CYP1A2ADORA2AADORA1AR
SCHEMBL28854068 0.74 ADA (0.31) KAT2B
SCHEMBL30119632 0.72 CYP17A1 (0.60) CYP17A1CYP1A2ADORA2AADORA1AR
SCHEMBL31363591 0.67 CYP17A1 (0.51) CYP17A1CYP1A2AR
SCHEMBL903225 0.66 CYP17A1 (0.70) CYP17A1CYP1A2
SCHEMBL38662718 0.65 TDP1 (0.63) FDPS
SCHEMBL28634932 0.64 CYP17A1 (0.48) CYP17A1CYP1A2AR
SCHEMBL27896288 0.64 TERT (0.40) KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429410-A Polyheterocyclic substituted pyrimidine or pyridylamine derivatives, compositions and medical uses thereof 上海海雁医药科技有限公司 2021-09-24 CN disclosed