SCHEMBL28645790

SCHEMBL28645790

CCn1c(=O)c(Br)cn(CC(=O)OC)c1=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 2/20 0.42
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.37
GAA P10253 1/20 0.36
ASAH1 Q13510 1/20 0.36
TNF P01375 2/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28926290 0.89 CDK9 (0.43) CDK9SMN1; SMN2KDM4EGAAASAH1
SCHEMBL28652315 0.85 CDK9 (0.42) CDK9SMN1; SMN2KDM4EGAAASAH1
SCHEMBL28638729 0.85 CDK9 (0.42) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28646718 0.83 CDK9 (0.41) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL21900263 0.83 CDK9 (0.44) CDK9KDM4EKMT2AALDH1A1POLB
SCHEMBL28639222 0.82 CDK9 (0.40) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28660748 0.82 SMN1; SMN2 (0.51) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28644072 0.81 CDK9 (0.40) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28652146 0.81 CDK9 (0.40) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28657237 0.80 CDK9 (0.39) CDK9SMN1; SMN2KDM4EKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3708566-B1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RES & DEV (FR) 2023-02-08 EP disclosed
CN-107428744-B Novel heterocyclic compounds and their use in medicine and cosmetics 盖尔德马研究及发展公司 2021-09-24 CN disclosed