SCHEMBL28652146

SCHEMBL28652146

COC(=O)Cn1cc(Br)c(=O)n(CCS(C)(=O)=O)c1=O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.38
KDM4E B2RXH2 3/20 0.37
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 1/20 0.32
KAT2B Q92831 1/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
TNF P01375 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28651448 0.86 SMN1; SMN2 (0.39) SMN1; SMN2KDM4ENPC1RAB9AMEN1
SCHEMBL28926290 0.84 CDK9 (0.43) CDK9SMN1; SMN2KDM4EGAACYP2C9
SCHEMBL28638729 0.83 CDK9 (0.42) CDK9SMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL28646718 0.82 CDK9 (0.41) CDK9SMN1; SMN2KDM4EMAPTMEN1
SCHEMBL28645790 0.81 CDK9 (0.44) CDK9SMN1; SMN2KDM4EKMT2AGAA
SCHEMBL28639222 0.81 CDK9 (0.40) CDK9SMN1; SMN2KDM4EMAPTMEN1
SCHEMBL19874000 0.80 ALDH1A1 (0.34) CDK9TNFALDH1A1
SCHEMBL28644072 0.80 CDK9 (0.40) CDK9SMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL28651571 0.79 CDK9 (0.39) CDK9SMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL28660748 0.78 SMN1; SMN2 (0.51) CDK9SMN1; SMN2KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428744-B Novel heterocyclic compounds and their use in medicine and cosmetics 盖尔德马研究及发展公司 2021-09-24 CN disclosed