SCHEMBL28647264

SCHEMBL28647264

Cn1nc(COc2ccc(N3CCN(C(=O)OC(C)(C)C)C(C(C)(C)C)C3)cc2)c(Br)c1CO

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 13/20 0.39
GPR119 Q8TDV5 3/20 0.37
NPC1 O15118 2/20 0.36
LMNA P02545 1/20 0.36
NR2F2 P24468 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NR1H3 Q13133 12/20 0.34
ESRRB O95718 1/20 0.34
ESR1 P03372 1/20 0.34
ESRRA P11474 1/20 0.34
ESRRG P62508 1/20 0.34
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28643152 0.85 NR1H2 (0.38) NR1H2GPR119NPC1LMNANR2F2
SCHEMBL19635047 0.85 SMN1; SMN2 (0.47) GPR119NPC1LMNANR2F2HTT
SCHEMBL21802247 0.78 MAPT (0.44) NPC1LMNASMN1; SMN2
SCHEMBL29291172 0.74 NR1H2 (0.53) NR1H2GPR119LMNANR1H3
SCHEMBL19634868 0.72 SMN1; SMN2 (0.47) GPR119NPC1LMNANR2F2HTT
SCHEMBL19615367 0.72 MEN1 (0.44) LMNAHTTSMN1; SMN2
SCHEMBL23251241 0.71 SMN1; SMN2 (0.46) GPR119NPC1LMNANR2F2HTT
SCHEMBL19635767 0.70 SMN1; SMN2 (0.45) GPR119NPC1LMNANR2F2HTT
SCHEMBL28956431 0.69 NR1H2 (0.54) NR1H2GPR119LMNAHTTNR1H3
SCHEMBL31180987 0.69 GPR119 (0.59) NR1H2GPR119NPC1NR1H3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715632-B Macrocyclic indole derivatives 拜尔公开股份有限公司 2021-10-26 CN disclosed