SCHEMBL28648256

SCHEMBL28648256

Cn1cc(-c2cccc(C(F)(F)F)n2)c(C=O)n1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.40
IDH1 O75874 8/20 0.39
IDH2 P48735 1/20 0.39
CSNK1D P48730 1/20 0.38
CSNK1E P49674 1/20 0.38
HCRTR1 O43613 1/20 0.38
NOTUM Q6P988 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
GRIN2B Q13224 1/20 0.34
MBOAT4 Q96T53 1/20 0.34
COMT P21964 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16321221 0.80 ALDH1A1 (0.44) TGFBR1IDH1IDH2CSNK1DCSNK1E
SCHEMBL19207002 0.77 HCRTR1 (0.47) TGFBR1IDH1IDH2CSNK1DCSNK1E
SCHEMBL28658603 0.73 BRD4 (0.48) TGFBR1
SCHEMBL19806307 0.70 NOTUM (0.42) TGFBR1IDH1IDH2CSNK1DCSNK1E
SCHEMBL19806523 0.70 GABRA1 (0.47) TGFBR1IDH1IDH2NOTUMGABRA1
SCHEMBL20028677 0.69 TGFBR1 (0.47) TGFBR1CSNK1DCSNK1ENOTUMGRIN2B
SCHEMBL16399255 0.69 HTR2B (0.48) IDH1IDH2NOTUMGABRA1GABRG2
SCHEMBL31003055 0.68 NOTUM (0.38) TGFBR1IDH1IDH2NOTUMGABRA1
SCHEMBL29320448 0.68 NOTUM (0.38) TGFBR1IDH1IDH2NOTUMGABRA1
SCHEMBL16116264 0.68 KMT2A (0.40) CSNK1DCSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109219606-B Halogen substituted piperidines as orexin receptor modulators 阿斯利康(瑞典)有限公司 2021-10-01 CN disclosed