SCHEMBL28649583

SCHEMBL28649583

COc1cc(C)oc(=O)c1CO

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
MEN1 O00255 3/20 0.45
MAPT P10636 3/20 0.45
KMT2A Q03164 3/20 0.45
PTGS1 P23219 6/20 0.44
PTGS2 P35354 6/20 0.44
USP2 O75604 1/20 0.44
CYP3A4 P08684 1/20 0.44
NQO1 P15559 2/20 0.43
KLK7 P49862 1/20 0.41
KLK5 Q9Y337 1/20 0.41
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
RECQL P46063 1/20 0.39
IDO1 P14902 2/20 0.38
BRAF P15056 1/20 0.38
ANTXR2 P58335 1/20 0.38
XDH P47989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6415919 0.71 CYP3A4 (0.50) KDM4EMEN1MAPTKMT2APTGS1
SCHEMBL8745776 0.67 NQO1 (0.59) KDM4EMEN1MAPTKMT2ANQO1
SCHEMBL12704738 0.67 MCL1 (0.40) KDM4EMEN1KMT2ACYP3A4
SCHEMBL1047858 0.66 ALDH1A1 (0.46) USP2CYP3A4
SCHEMBL31207104 0.66 CYP3A4 (0.56) MEN1MAPTKMT2APTGS1PTGS2
SCHEMBL29092099 0.66 MCL1 (0.39) KDM4EMEN1MAPTKMT2AGAA
SCHEMBL1225856 0.66 ACHE (0.46) KDM4EMAPT
SCHEMBL11860188 0.66 KDM4E (0.40) KDM4EMEN1MAPTKMT2APTGS1
SCHEMBL11131991 0.65
SCHEMBL21776517 0.65 MCL1 (0.38) KDM4EMEN1KMT2ACYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108913731-B Pyran compound with immunosuppressive activity and preparation method and application thereof 海南大学 2021-11-16 CN disclosed
CN-108913731-A A kind of pyran compounds and its preparation method and application with immunosuppressive activity 海南大学 2018-11-30 CN disclosed