SCHEMBL28653645

SCHEMBL28653645

CC(C)(C)OC(=O)Nc1ccc(C(=O)CBr)cn1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.53
HDAC1 Q13547 1/20 0.45
BCL2 P10415 1/20 0.45
NAMPT P43490 3/20 0.41
GSK3B P49841 3/20 0.41
DYRK1A Q13627 1/20 0.41
DEGS1 O15121 1/20 0.40
ATR Q13535 1/20 0.40
HCAR3 P49019 4/20 0.38
MAPKAPK2 P49137 1/20 0.38
CYP17A1 P05093 1/20 0.38
AKT1 P31749 1/20 0.38
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15059736 0.88 GRIN2B (0.53) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL14652137 0.88 GRIN2B (0.53) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL30320778 0.86 GSK3B (0.46) HDAC1GSK3BDEGS1HCAR3EPHX2
SCHEMBL25702957 0.86 GSK3B (0.46) HDAC1GSK3BDEGS1HCAR3EPHX2
SCHEMBL13838587 0.85 GRIN2B (0.52) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL29651977 0.83 HCAR3 (0.57) GRIN2BHDAC1BCL2HCAR3
SCHEMBL2877186 0.83 HCAR3 (0.57) GRIN2BHDAC1BCL2HCAR3
SCHEMBL28658285 0.83 GRIN2B (0.48) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL31727242 0.83 GRIN2B (0.48) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL30552385 0.82 HDAC1 (0.51) GRIN2BHDAC1BCL2NAMPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527261-A Pyridone or pyrimidone derivative and preparation method and application thereof 浙江海正药业股份有限公司 2021-10-22 CN disclosed