SCHEMBL28658285

SCHEMBL28658285

CC(=O)c1ccc(NC(=O)OC(C)(C)C)nc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.48
HDAC1 Q13547 1/20 0.46
BCL2 P10415 2/20 0.45
NAMPT P43490 2/20 0.44
CYP17A1 P05093 2/20 0.44
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
DEGS1 O15121 2/20 0.43
HCAR3 P49019 2/20 0.41
BECN1 Q14457 1/20 0.41
PTK2 Q05397 1/20 0.41
NNMT P40261 1/20 0.41
ATR Q13535 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31727242 1.00 GRIN2B (0.48) GRIN2BHDAC1BCL2NAMPTCYP17A1
SCHEMBL31599569 0.88 GRIN2B (0.47) GRIN2BHDAC1BCL2NAMPTCYP17A1
SCHEMBL13876322 0.88 GRIN2B (0.47) GRIN2BHDAC1BCL2NAMPTCYP17A1
SCHEMBL2877186 0.88 HCAR3 (0.57) GRIN2BHDAC1BCL2HCAR3
SCHEMBL29651977 0.88 HCAR3 (0.57) GRIN2BHDAC1BCL2HCAR3
SCHEMBL7936803 0.87 HCAR3 (0.55) GRIN2BHDAC1BCL2HCAR3
SCHEMBL5734042 0.87 NNMT (0.58) GRIN2BHDAC1BCL2NAMPTGSK3B
SCHEMBL2772417 0.87 MAPK1 (0.51) GRIN2BHDAC1BCL2NAMPTCYP17A1
Lithium Ion SCHEMBL7936799 0.85 GRIN2B (0.47) GRIN2BHDAC1BCL2NAMPTCYP17A1
SCHEMBL20828520 0.85 GRIN2B (0.47) GRIN2BHDAC1BCL2NAMPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527261-A Pyridone or pyrimidone derivative and preparation method and application thereof 浙江海正药业股份有限公司 2021-10-22 CN disclosed