SCHEMBL28655154

SCHEMBL28655154

NC(=O)N(c1cccc(C(F)(F)F)c1)c1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
RORC P51449 1/20 0.37
RORB Q92753 1/20 0.37
KDR P35968 1/20 0.37
KIF11 P52732 2/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
EPHX1 P07099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27653563 0.87 P2RX1 (0.41) CES2MEN1KMT2AALDH1A1RORC
SCHEMBL5606524 0.86 CES2 (0.50) CES2MEN1KMT2AALDH1A1KIF11
SCHEMBL3674538 0.85 CES2 (0.40) CES2MEN1KMT2AALDH1A1RORC
SCHEMBL28217598 0.82 PTGIR (0.46) CES2MEN1KMT2AKIF11HTR3E
SCHEMBL7609002 0.78 SRD5A2 (0.55) CES2MEN1KMT2AALDH1A1HTT
SCHEMBL7739130 0.78 CES2 (0.50) CES2MEN1KMT2AALDH1A1LMNA
SCHEMBL4246399 0.77 HTR3E (0.49) MEN1KMT2AKDRHTR3EHTR3B
SCHEMBL7738559 0.77 SRD5A2 (0.52) CES2MEN1KMT2AALDH1A1LMNA
SCHEMBL28217604 0.77 GRM4 (0.44) MEN1KMT2AALDH1A1KDRHTR3E
SCHEMBL1942998 0.76 POLQ (0.41) KMT2AALDH1A1KDRLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113574055-A PCSK9 inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2021-10-29 CN disclosed