SCHEMBL286558

SCHEMBL286558

N#Cc1ccc2c(c1)C=COC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
PNMT P11086 6/20 0.39
DRD2 P14416 4/20 0.39
DRD3 P35462 4/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
KDM1A O60341 2/20 0.34
CYP2A6 P11509 1/20 0.33
PDE4B Q07343 2/20 0.31
CHRM1 P11229 1/20 0.31
PDE4A P27815 1/20 0.31
ADRA1A P35348 1/20 0.31
PDE1A P54750 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE7A Q13946 1/20 0.31
PDE3A Q14432 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29740368 0.72 CA1 (0.44) TRPA1PNMTDRD2DRD3CA12
SCHEMBL148119 0.72 CA1 (0.44) TRPA1PNMTDRD2DRD3CA12
SCHEMBL29740370 0.72 CA1 (0.44) TRPA1PNMTDRD2DRD3CA12
Hydrochloric Acid SCHEMBL20919478 0.70 CA1 (0.43) TRPA1PNMTDRD2DRD3CA12
SCHEMBL15320222 0.69 PNMT (0.43) TRPA1PNMTDRD2DRD3CA12
SCHEMBL3296947 0.68 DRD2 (0.42) TRPA1PNMTDRD2DRD3CA12
SCHEMBL6739755 0.68
SCHEMBL31545183 0.67 PNMT (0.48) TRPA1PNMTDRD2DRD3KDM1A
SCHEMBL2809825 0.67 PNMT (0.48) TRPA1PNMTDRD2DRD3KDM1A
Hydrochloric Acid SCHEMBL7003642 0.67 PARP1 (0.50) TRPA1PNMTDRD2DRD3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427444-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2012-03-14 EP disclosed