SCHEMBL28656240

SCHEMBL28656240

CC(=O)OC(=CCc1cccc(Cl)c1)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.43
MAOA P21397 3/20 0.41
HCAR2 Q8TDS4 1/20 0.39
GRM5 P41594 1/20 0.39
TRPV1 Q8NER1 1/20 0.38
EPHX2 P34913 1/20 0.38
RIPK1 Q13546 1/20 0.38
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
CTBP2 P56545 1/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29718860 0.85 MAOB (0.40) MAOBMAOACTBP2POLB
SCHEMBL28670520 0.83 CES1 (0.42) MAOB
SCHEMBL28653905 0.79 CYP1A2 (0.38)
SCHEMBL28418613 0.78 HCAR2 (0.39) MAOBHCAR2TRPV1EPHX2HTR3E
SCHEMBL28929352 0.77 TRPA1 (0.50) MAOBMAOARIPK1
SCHEMBL28654237 0.76 TRPA1 (0.38) MAOB
SCHEMBL28664225 0.76 RXRA (0.36) RXRARXRBPOLB
SCHEMBL28650409 0.76 MMP12 (0.39)
SCHEMBL28670280 0.75 MAOB (0.43) MAOB
SCHEMBL28658852 0.75 TRPA1 (0.37) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354586-B Preparation method of trifluoromethyl-containing pyrazolone compound 大连理工大学 2022-06-10 CN disclosed
CN-113717092-A Preparation method of trifluoromethyl-containing 3-substituted-2-indolinone compound 美罗药业股份有限公司 2021-11-30 CN disclosed
CN-113354586-A Preparation method of trifluoromethyl-containing pyrazolone compound 大连理工大学 2021-09-07 CN disclosed