SCHEMBL28656241

SCHEMBL28656241

O=C(O)c1cc2cccsc-2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 1/20 0.46
KMO O15229 1/20 0.46
SRPK1 Q96SB4 1/20 0.45
RPS6KB2 Q9UBS0 1/20 0.45
DAO P14920 1/20 0.45
DHODH Q02127 2/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 1/20 0.43
PTPN1 P18031 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
EGLN1 Q9GZT9 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC2 Q92769 1/20 0.42
HTR1A P08908 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CCKAR P32238 1/20 0.42
HTR5A P47898 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31222146 0.85 KAT6A (0.57) KAT6AKMOSRPK1RPS6KB2KDM4E
SCHEMBL940399 0.85 KAT6A (0.57) KAT6AKMOSRPK1RPS6KB2KDM4E
SCHEMBL9637810 0.78 PTPN1 (0.48) KAT6ASRPK1RPS6KB2DAOKDM4E
SCHEMBL3915007 0.78 TPMT (0.50) KAT6ASRPK1RPS6KB2DHODHKDM4E
Benzoic Acid SCHEMBL26966093 0.77 DAO (0.54) KAT6AKMODAOKDM4EMAPT
SCHEMBL27623947 0.76 KAT6A (0.55) KAT6AHDAC1HDAC3HDAC2HTR1A
SCHEMBL27905638 0.75 KAT6A (0.58) KAT6AKMOHDAC1HDAC3HDAC2
SCHEMBL938500 0.74 KMO (0.52) KMODAODHODHKDM4EMEN1
SCHEMBL420705 0.74 KDM4E (0.55) SRPK1RPS6KB2DAOKDM4EMAPT
SCHEMBL6040460 0.74 KAT6A (0.47) KAT6AKMOSRPK1RPS6KB2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108976172-B 4-pyrimidinediamine micromolecule organic compound and derivative and application thereof 华东师范大学 2021-12-07 CN disclosed