SCHEMBL7936803

SCHEMBL7936803

CC(C)(C)OC(=O)Nc1ccc(C(=O)O)cn1.[LiH]

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 17/20 0.55
GRIN2B Q13224 1/20 0.50
HCAR2 Q8TDS4 2/20 0.48
BCL2 P10415 1/20 0.47
HDAC1 Q13547 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29651977 0.98 HCAR3 (0.57) HCAR3GRIN2BHCAR2BCL2HDAC1
SCHEMBL2877186 0.98 HCAR3 (0.57) HCAR3GRIN2BHCAR2BCL2HDAC1
SCHEMBL5543076 0.87 BCL2 (0.52) HCAR3GRIN2BBCL2HDAC1
SCHEMBL28658285 0.87 GRIN2B (0.48) HCAR3GRIN2BBCL2HDAC1
SCHEMBL31727242 0.87 GRIN2B (0.48) HCAR3GRIN2BBCL2HDAC1
SCHEMBL2772417 0.85 MAPK1 (0.51) HCAR3GRIN2BBCL2HDAC1
SCHEMBL5734042 0.85 NNMT (0.58) GRIN2BBCL2HDAC1
SCHEMBL31599569 0.84 GRIN2B (0.47) HCAR3GRIN2BBCL2HDAC1
SCHEMBL20828520 0.84 GRIN2B (0.47) HCAR3GRIN2BBCL2HDAC1
SCHEMBL2058148 0.84 HCAR3 (0.54) HCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed