SCHEMBL28658384

SCHEMBL28658384

COC(=O)NC1(c2cccc(Br)c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
FAAH O00519 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
GAA P10253 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HCAR3 P49019 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
MAPT P10636 2/20 0.38
CYP1A2 P05177 1/20 0.38
RECQL P46063 1/20 0.38
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31360210 0.86 CTSB (0.40) FAAHTRPV1GAANPSR1ALDH1A1
SCHEMBL2036519 0.86 CTSB (0.40) FAAHTRPV1GAANPSR1ALDH1A1
SCHEMBL2030447 0.83 NPSR1 (0.44) HDAC3HDAC1HDAC2HDAC6FAAH
SCHEMBL28647793 0.82 HDAC3 (0.48) HDAC3HDAC1HDAC2HDAC6FAAH
SCHEMBL30344979 0.82 RAB9A (0.43) GAANPSR1ALDH1A1SMN1; SMN2MAPT
SCHEMBL31292775 0.81 AKT1 (0.41) FAAHTRPV1GAANPSR1ALDH1A1
SCHEMBL30749325 0.81 AKT1 (0.43) FAAHTRPV1GAANPSR1ALDH1A1
SCHEMBL14672673 0.81 GAA (0.41) HDAC3HDAC1HDAC2HDAC6FAAH
SCHEMBL22470395 0.81 GAA (0.35) HDAC3HDAC1HDAC2HDAC6FAAH
SCHEMBL27853653 0.80 OPRM1 (0.49) HDAC3HDAC1HDAC2HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113631538-A Novel potassium channel inhibitors 萨尼奥纳有限责任公司 2021-11-09 CN claimed
CN-113631538-A Novel potassium channel inhibitors 萨尼奥纳有限责任公司 2021-11-09 CN disclosed