Miconazole

Miconazole

SCHEMBL2866

Clc1ccc(COC(Cn2ccnc2)c2ccc(Cl)cc2Cl)c(Cl)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Miconazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 12/20 1.00
CYP2C9 P11712 7/20 1.00
CYP3A4 P08684 6/20 1.00
LMNA P02545 5/20 1.00
CYP1A2 P05177 5/20 1.00
CYP2D6 P10635 5/20 1.00
CYP2C19 P33261 5/20 1.00
NR1I2 O75469 4/20 1.00
NR3C1 P04150 4/20 1.00
CYP17A1 P05093 4/20 1.00
PGR P06401 4/20 1.00
ADRB1 P08588 4/20 1.00
ADORA3 P0DMS8 4/20 1.00
DRD2 P14416 4/20 1.00
SLC6A2 P23975 4/20 1.00
SLC6A4 P31645 4/20 1.00
OPRK1 P41145 4/20 1.00
SLC6A3 Q01959 4/20 1.00
KCNH2 Q12809 4/20 1.00
CHRM3 P20309 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Miconazole SCHEMBL9662051 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
(R)-Miconazole SCHEMBL2867 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
(R)-Miconazole SCHEMBL30594078 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
Miconazole SCHEMBL64342 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
Miconazole SCHEMBL13934598 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
Miconazole SCHEMBL7647866 1.00 IDO1 (1.00) IDO1CYP2C9CYP3A4LMNACYP1A2
(R)-Miconazole SCHEMBL3131763 0.99 IDO1 (0.98) IDO1CYP2C9CYP3A4LMNACYP1A2
(R)-Miconazole SCHEMBL10575725 0.99 IDO1 (0.98) IDO1CYP2C9CYP3A4LMNACYP1A2
Miconazole SCHEMBL9479815 0.99 IDO1 (0.98) IDO1CYP2C9CYP3A4LMNACYP1A2
Miconazole SCHEMBL10575722 0.99 IDO1 (0.98) IDO1CYP2C9CYP3A4LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 50053 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107113-A1 MODIFIED CELLS FOR PROGRAMMING EXTRA ENVELOPED VIRUSES (EEVs) AND THEIR USE FOR PRODUCING THE EEVs, THE PROGRAMMED EEVs AND USES THEREOF CALIDI BIOTHERAPEUTICS (NEVADA), INC. (US) 2026-05-21 WO claimed
WO-2026106952-A1 METHODS FOR TREATING CONGENITAL DISORDERS OF GLYCOSYLATION CDG CARE (US) 2026-05-21 WO claimed
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
WO-2026102345-A1 METHODS OF ADMINISTERING THE VOLTAGE-GATED POTASSIUM CHANNEL OPENER AZETUKALNER XENON PHARMACEUTICALS INC. (CA) 2026-05-15 WO claimed
US-20260124224-A1 USE OF COMBINED COMPOSITION IN PREPARING DRUG FOR RESISTING FUNGAL AND BACTERIAL INFECTIONS NATIONAL CENTER FOR NANOSCIENCE AND TECHNOLOGY (CN) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
US-20260115192-A1 PHARMACEUTICAL COMPOSITIONS SHENZHEN PHARMACIN CO LTD (CN) 2026-04-30 US claimed
EP-3222270-B1 COMPOSITIONS FOR MUCOSAL ADHESION AND USES THEREOF BIONANOPLUS S L (ES) 2026-04-29 EP claimed
US-20260102419-A1 USE OF COMPOUNDS IN THE TREATMENT OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH) 2026-04-16 US claimed
US-4427660-A Formyl-methionyl chemotatic peptide antibiotic conjugates useful in treating infections RESEARCH CORPORATION (US) 1984-01-24 US claimed
EP-0098743-A1 Phenyl alpha-acyloxyacetamide derivates and their therapeutic use Yu, Ruey J., Dr. (US) 1984-01-18 EP claimed
EP-0094329-A1 Tanning process for rendering leathers mycostatic, antimycosic and antifungicidal, and articles produced thereby Roux, Joel (FR) 1983-11-16 EP claimed
EP-0053936-A2 Surgical dressing Johnson & Johnson Products Inc. (US) 1982-06-16 EP claimed
US-4321257-A Potentiated medicaments JOHNSON & JOHNSON (US) 1982-03-23 US claimed
US-4294852-A WATER, AN ALIPHATIC ALCOHOL AND AN ORGANIC ACID TO ADJUST THE PH OF THE VEHICLE JOHNSON & JOHNSON (US) 1981-10-13 US claimed
US-4277475-A FOR BOTH MALES AND FEMALES SYNTEX (U.S.A.) INC. (US) 1981-07-07 US claimed
US-4247552-A Contraceptive compositions and methods employing 1-substituted imidazole derivatives SYNTEX (U.S.A.) INC. (US) 1981-01-27 US claimed
US-4197318-A CYCLOHEXYL SUBSTITUTED ALKANOLS AS POTENTIATORS JOHNSON & JOHNSON (US) 1980-04-08 US claimed
US-4082881-A STEROIDS, DERMATITIS E. R. SQUIBB & SONS, INC. (US) 1978-04-04 US claimed