SCHEMBL28660397

SCHEMBL28660397

Cc1nc(-c2ccnc(C#N)c2)sc1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.56
XDH P47989 7/20 0.56
TARBP2 Q15633 2/20 0.55
ABCC4 O15439 1/20 0.55
ABCB11 O95342 1/20 0.55
PGR P06401 1/20 0.55
CHRM1 P11229 1/20 0.55
PDE4A P27815 1/20 0.55
BLVRB P30043 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
ABCG2 Q9UNQ0 1/20 0.55
KDM4E B2RXH2 4/20 0.55
RAB9A P51151 3/20 0.55
GAA P10253 1/20 0.55
NPC1 O15118 1/20 0.52
POLB P06746 1/20 0.52
ALDH1A1 P00352 1/20 0.51
KMT2A Q03164 1/20 0.50
MYC P01106 1/20 0.45
GSK3B P49841 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28672541 0.84 CDC7 (0.65) XDHTARBP2ABCC4ABCB11PGR
SCHEMBL28653714 0.84 XDH (0.43) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL28677825 0.82 SMN1; SMN2 (0.44) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL28660406 0.80 SMN1; SMN2 (0.60) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL28672534 0.79 SMN1; SMN2 (0.63) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL28658387 0.79 SMN1; SMN2 (0.58) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL28660331 0.79 SMN1; SMN2 (0.49) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL27875453 0.78 CDC7 (0.63) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL19523322 0.77 XDH (0.63) SMN1; SMN2XDHTARBP2ABCC4ABCB11
SCHEMBL438271 0.77 XDH (0.68) SMN1; SMN2XDHTARBP2ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024534-B 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2023-03-21 CN claimed
CN-113024534-A 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2021-06-25 CN claimed
CN-113024534-B 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2023-03-21 CN disclosed
CN-113024534-A 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2021-06-25 CN disclosed